Antimalarial, Plasmodium falciparum, N-Alkylated Pyridinium Dimer, chloroquine-sensetive, Structure-Activity-RelationshipExploitation for New Antimalarials2000.01Pyridazine,Chemiluminescence,LuminolSynthesis of Pyridazine Derivatives and their Chemiluminescent Activity1993.01Development of New Analitical Reagent utilizing its Chemilumineseent Activity1993.01Heterocyclic Compound,Photocyclization,Structure-Activity RelationshipSynthesis of Novel Polycyclic Heterocyclic Compounds via Photocyclization and Evaluation of their Biological Activity1991.01 

Photograph

Name

SASAKI Kenji

Affiliation

Institute for Education and Student Services

Title

Professor

Sex

male

Research areas, keyword

Organic Chemistry, Drug Molecular Design, Structure-Activity-Relationship

Research Subject 【 display / non-display

  • Subject:Exploitation for New Antimalarials

    Object:

  • Subject:Synthesis of Pyridazine Derivatives and their Chemiluminescent Activity

  • Subject:Development of New Analitical Reagent utilizing its Chemilumineseent Activity

 
 

Research Achievement (Published Thesis) 【 display / non-display

  • Subject:Quercetin diacylglycoside analogues showing dual inhibition of DNA gyrase and topoisomerase IV as novel antibacterial agents (共著)

    Language:English

    Kind of Publishing:Academic Journal

    Journal name:Journal of Medicinal Chemistry , vol.54 (11) (p.3686 - 3703)

    Publish date:2011.11

    Author:「Hossion Abugafar M L」「Zamami Yoshito」「Kandahary Rafiya K」「Tsuchiya Tomofusa」「Ogawa Wakano」「Iwado Akimasa」「Sasaki Kenji」

    Co-writerThe multiple authorship

    DOI:10.1021/jm200010x

  • Subject:Design, synthesis, and biological evaluation of a novel series of quercetin diacylglucosides as potent anti-MRSA and anti-VRE agents (共著)

    Language:English

    Kind of Publishing:Academic Journal

    Journal name:Bioorganic & Medicinal Chemistry Letters , vol.20 (17) (p.5349 - 5352)

    Publish date:2010.09

    Author:「Hossion Abugafar M L」「Otsuka Nao」「Kandahary Rafiya K」「Tsuchiya Tomofusa」「Ogawa Wakano」「Iwado Akimasa」「Zamami Yoshito」「Sasaki Kenji」

    Co-writerThe multiple authorship

    DOI:10.1016/j.bmcl.2010.02.060

  • Subject:Pyridinium cationic-dimer antimalarials, unlike chloroquine, act selectively between the schizont stage and the ring stage of Plasmodium falciparum

    Language:

    Kind of Publishing:

    Journal name:Bioorganic & Medicinal Chemistry , vol.16 (11) (p.6027 - 6033)

    Publish date:2008.06

    Author:Mai Yoshikawa, Kazunori Motoshima, Kanji Fujimoto, Akihiro Tai, Hiroki Kakuta, *Kenji Sasaki

    Co-writerThe multiple authorship

  • Subject:Polycyclic N-Heterocyclic Compounds. Part 86: Synthesis and Evaluation of Antiplatelet Aggregation Activity of 2,4-Disubstituted 9-Chloro-5,6-dihydropyrimido[5,4-d]benzazepine and Related Compounds

    Language:English

    Kind of Publishing:Academic Journal

    Journal name:Journal of Heterocyclic Chemistry , vol.52 (3) (p.780 - 792)

    Publish date:2015.05

    Author:Kensuke Okuda, Shigeki Takarada, Takashi Hirota, Kenji Sasaki

    Co-writerThe multiple authorship

    DOI:10.1002/jhet.2190

  • Subject:Polycyclic N-Heterocyclic Compounds. Part 85: Synthesis and Evaluation of Antiplatelet Aggregation Activity of 2,4-Disubstituted 5,6-Dihydro[1]benzazepino[5,4-d]pyrimidine and Related Compounds

    Language:English

    Kind of Publishing:Academic Journal

    Journal name:Journal of Heterocyclic Chemistry , vol.52 (3) (p.888 - 895)

    Publish date:2015.05

    Author:Kensuke Okuda, Ying-Xue Zhang, Takashi Hirota, Kenji Sasaki

    Co-writerThe multiple authorship

    DOI:10.1002/jhet.2040

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